SURPASS-3 Trial: Tirzepatide vs Insulin Degludec — Superior Glucose Control With Weight Loss Instead of Gain

Medically reviewed by Dr. James Whitfield, DO, FACOI

The SURPASS-3 trial, published in The Lancet in 2021 by Ludvik et al., compared tirzepatide against insulin degludec in 1,444 patients with type 2 diabetes. The results were striking: tirzepatide 15mg reduced HbA1c by 2.37% with 12.9kg weight loss, while insulin degludec reduced HbA1c by only 1.34% with 2.3kg weight gain — a 15.2kg difference in body weight.

SURPASS-3: Rewriting the Insulin Paradigm

For decades, insulin has been the cornerstone of type 2 diabetes treatment when oral medications fail. The SURPASS-3 trial, published in The Lancet in October 2021 by Ludvik et al., challenged this paradigm by demonstrating that tirzepatide not only matched but dramatically exceeded insulin degludec in glycemic control — while producing massive weight loss instead of the weight gain that plagues insulin therapy [1].

Study Design

SURPASS-3 was a 52-week, open-label, randomized Phase 3 trial conducted at 122 sites across 13 countries. It enrolled 1,444 adults with type 2 diabetes inadequately controlled on metformin with or without an SGLT2 inhibitor.

Randomization (1:1:1:1):

  • Tirzepatide 5 mg weekly
  • Tirzepatide 10 mg weekly
  • Tirzepatide 15 mg weekly
  • Insulin degludec (titrated to fasting glucose <90 mg/dL)
  • Insulin degludec (Tresiba) was chosen as the comparator because it represents a modern, long-acting basal insulin with a favorable safety profile and low hypoglycemia risk — making it a strong comparator [1].

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    Glycemic Control: Tirzepatide Dominates

    Mean HbA1c Change from Baseline (~8.2%):

  • Tirzepatide 5 mg: -1.93%
  • Tirzepatide 10 mg: -2.20%
  • Tirzepatide 15 mg: -2.37%
  • Insulin degludec: -1.34%
  • Treatment Difference vs. Insulin (15 mg): -1.04% (P<0.001)

    HbA1c Target Achievement:

  • HbA1c <7.0%: 82% (5 mg), 90% (10 mg), 93% (15 mg) vs. 61% (insulin)
  • HbA1c <5.7%: 26% (5 mg), 39% (10 mg), 48% (15 mg) vs. 5% (insulin)
  • The fact that tirzepatide achieved nearly a full percentage point more HbA1c reduction than optimally titrated insulin is remarkable. Insulin has long been considered the most potent glucose-lowering therapy, yet tirzepatide surpassed it decisively [1].

    The Weight Story: Loss vs. Gain

    The weight data represents the most dramatic contrast:

    Mean Body Weight Change:

  • Tirzepatide 5 mg: -7.5 kg (-7.5%)
  • Tirzepatide 10 mg: -10.7 kg (-10.7%)
  • Tirzepatide 15 mg: -12.9 kg (-12.9%)
  • Insulin degludec: +2.3 kg (+2.4%)
  • Total Weight Difference (15 mg vs. insulin): 15.2 kg (33.5 lbs)

    This 15.2 kg difference is clinically enormous. A patient choosing tirzepatide over insulin would weigh approximately 33 pounds less after one year — while achieving better glucose control [1].

    Why Insulin Causes Weight Gain

    Understanding why insulin promotes weight gain helps explain tirzepatide's advantage:

  • Anabolic effects: Insulin promotes fat storage and inhibits fat breakdown
  • Hypoglycemia avoidance: Patients eat defensively to prevent low blood sugar
  • Reduced glucosuria: Better glucose control means less glucose lost in urine (fewer "free" calories excreted)
  • Appetite stimulation: Insulin can increase hunger through central nervous system effects
  • Tirzepatide avoids all of these mechanisms while providing superior glucose lowering through appetite reduction, improved insulin sensitivity, and glucose-dependent insulin secretion [2].

    Safety Comparison

    Hypoglycemia (<54 mg/dL):

  • Tirzepatide: 0.4-1.1%
  • Insulin degludec: 7.5%
  • The dramatically lower hypoglycemia rate with tirzepatide is a major safety advantage. Hypoglycemia is the most feared complication of insulin therapy, limiting dose titration and causing significant anxiety.

    Gastrointestinal Events:

  • Nausea: 12-24% (tirzepatide) vs. 2% (insulin)
  • Diarrhea: 15-17% vs. 4%
  • These were the main adverse events more common with tirzepatide
  • Discontinuation due to AEs:

  • Tirzepatide: 3-7%
  • Insulin: 1% [1]
  • Liver Fat Reduction

    A notable secondary finding was tirzepatide's effect on liver fat:

  • Tirzepatide reduced liver fat content by 33-37% (measured by MRI)
  • Insulin degludec reduced liver fat by only 8%
  • This has implications for non-alcoholic fatty liver disease (NAFLD), which affects the majority of patients with type 2 diabetes
  • Clinical Implications

    SURPASS-3 has several practice-changing implications:

  • Insulin delay: Tirzepatide provides a powerful alternative before starting insulin
  • Insulin replacement: Some patients currently on insulin may benefit from switching to tirzepatide
  • Weight management: Eliminates the weight gain dilemma of insulin therapy
  • Simplified regimen: Once-weekly injection vs. daily insulin (often multiple daily injections)
  • Hypoglycemia reduction: Dramatically lower risk of dangerous low blood sugar
  • > Related Comparison: MOTS-C vs Metformin: Metabolic Comparison

    > Related Comparison: Ozempic vs Mounjaro: Complete Comparison

    References

  • Ludvik B, Giorgino F, Jódar E, et al. "Once-weekly tirzepatide versus once-daily insulin degludec as add-on to metformin with or without SGLT2 inhibitors in patients with type 2 diabetes (SURPASS-3): a randomised, open-label, parallel-group, phase 3 trial." The Lancet. 2021;398(10300):583-598. PubMed: 34370970
  • Nauck MA, D'Alessio DA. "Tirzepatide, a dual GIP/GLP-1 receptor co-agonist for the treatment of type 2 diabetes with unmatched effectiveness." Cardiovascular Diabetology. 2022;21:169. PubMed: 36050763
  • Heerspink HJL, Sattar N, Pavo I, et al. "Effects of tirzepatide versus insulin glargine on kidney outcomes in type 2 diabetes in the SURPASS-4 trial." The Lancet Diabetes & Endocrinology. 2022;10(11):774-785. PubMed: 36152639
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    Related Reading

    Explore more in-depth guides on related topics:

  • SURPASS-1 Trial: Tirzepatide Monotherapy Reduces HbA1c by 2.07% in Drug-Naive Type 2 Diabetes
  • SURMOUNT-2 Trial: Tirzepatide Delivers 15.7% Weight Loss in Adults With Obesity and Diabetes
  • SURMOUNT-1 Trial: Tirzepatide Achieves Up to 22.5% Weight Loss in Adults Without Diabetes
  • SURPASS-2 Trial: Tirzepatide Beats Semaglutide Head-to-Head in Type 2 Diabetes
  • SURPASS-4 Trial: Tirzepatide vs Insulin Glargine in High Cardiovascular Risk Patients
  • For a comprehensive overview, see our Complete Guide to Peptide Therapy. For a deeper dive into this area, see peptide monitoring blood panels.

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